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A highly facile single‐step synthetic approach to 3‐iodoquinolines has been developed for the first time from readily available 2‐aminobenzophenones and terminal alkynes. The reaction involves the nucleophilic addition of terminal alkynes to 2‐aminobenzophenones followed by a regioselective iodocyclization (6‐endo‐dig) to furnish 2,4‐disubstituted 3‐iodoquinolines in high yields. In general, 2,4‐diaryl‐substituted products were isolated without the need for column chromatography.

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Microwave Assisted, Ca(II)-Catalyzed Ritter Reaction for the Green Synthesis of Amides. -An efficient solvent-free synthesis of various primary amides from alcohols and nitriles through Cu-catalyzed Ritter reaction is presented. -(YARAGORLA*, S.; SINGH, G.; LAL SAINI, P.; REDDY, M. K.; Tetrahedron Lett. 55 (2014) 33, 4657-4660, http://dx.

Alkaline Earth Metal Catalyzed Cascade, One-Pot, Solvent-Free, and Scalable Synthesis of Pyranocoumarins and Benzo[b]pyrans. -(YARAGORLA*, S.; SAINI, P. L.; SINGH, G.; Tetrahedron Lett. 56 (2015) 13, 1649-1653, http://dx.

Facile multicomponent reactions for the synthesis of indolyl and oxindolyl acrylates as well as bisacrylates are presented.

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