Mechanism by Which 3-Enol Etherification Enhances the Oral Activity of Methyltestosterone in Rats

Meli, A; Honrath, W; Wolff, A.

doi:10.1210/endo-74-1-79

Search citation statements

Order By: Relevance

Paper Sections

Select...

Citation Types

Supporting

Mentioning

Contrasting

Year Published

1965

1971

Publication Types

Select...

Article4

Book3

Relationship

Self Cite1

Independent6

Authors

Journals

Cited by 9 publications

(2 citation statements)

References 0 publications

Supporting

Mentioning

Contrasting

Order By: Relevance

“…tivity is attributed to storage in, and a subsequent release from, body fat after administration (6,7 ) . This report describes the activity of quinestrol compared with estradiol-l7p on the pattern of estrogen withdrawal bleeding in the castrated rhesus monkey.…”

mentioning

confidence: 99%

Estrogenic Properties of Quinestrol and Estradiol-17 in the Ovariectomized Rhesus Monkey

Hisaw¹,

Mischler²,

Kroc³

1971

Experimental Biology and Medicine

View full text Add to dashboard Cite

mentioning

confidence: 99%

Estrogenic Properties of Quinestrol and Estradiol-17 in the Ovariectomized Rhesus Monkey

Hisaw¹,

Mischler²,

Kroc³

1971

Experimental Biology and Medicine

View full text Add to dashboard Cite

“…Though many studies on enol ether analogues of progesterone (2)(3)(4)(5)(6)(7) and certain androgens (2,7,(8)(9)(10)(11) have been reported, little is known about similar derivatives of 19-nortestosterone. Experiments with the 3-cyclopentyl enol ether of 17aethynyl-19-nortestosterone-l7p-acetate [ quingestanol acetate (QA)] showed that enol etherification generally enhances most biological activities as compared with its parent ketone (2,4,5,7,12).…”

mentioning

confidence: 99%