Design, Synthesis and Biological Activities Evaluation of N-(Substitutedbenzoyl)-N'-4,7-dimethoxy-[1,2,4]-triazolo[1,5-c]pyrimidine (Thio)ureas

Wei, Kailun; Jiang, Lin; Miao, Chengxia; Li, Ying

doi:10.6023/cjoc202003001

Cited by 1 publication

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“…The inhibition rate of compound 23 (Figure 7) on B. cinerea was 67.25% at 50 mg/L and the addition of electron-withdrawing groups to the benzene ring was conducive to enhancing the fungicidal activity of the compound [70]. The EC 50 value of compound 24 (Figure 8) for Gibberella zeae (G. zeae) was 24.8 mg/L [71].…”

Section: Antifungal Activitymentioning

confidence: 99%

Research progress of triazole derivatives in the discovery of agricultural chemicals

Song,

Wang,

Cai

et al. 2023

Journal of Heterocyclic Chem

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Triazole groups play an important role in the construction of agricultural bioactive molecules, often acting as linking units to organically graft different pharmacophore groups, so as to obtain efficient and broad‐spectrum pesticide molecules. After decades of development, triazole derivatives have made remarkable achievements in the discovery of pesticides, especially the discovery of fungicides. In addition, highly effective triazole insecticides, herbicides, and anti‐plant virus agents have also been found, and commercial triazole pesticides have occupied a large market share. At present, the study of triazole compounds has become one of the important fields in the development of new pesticides. We systematically reviewed the application of triazole derivatives in the discovery of new pesticides since 2010, summarized the antifungal, antibacterial, insecticidal, herbicidal, and anti‐plant virus activities of triazole derivatives, and discussed the structure–activity relationship and mechanism of action in order to provide inspiration and ideas for the discovery of new triazole agrochemicals.

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Section: Antifungal Activitymentioning

confidence: 99%