A Literature Review on Antipyrinein Chemistry Fields

Aljamali, Nagham Mahmood; Aati, Saba Abd Alhussain; Obaid, Nadia Hussein; Wannas, Fatimah A.

doi:10.46545/aijser.v2i1.41

Cited by 6 publications

(6 citation statements)

References 24 publications

Supporting

Mentioning

Contrasting

Order By: Relevance

“…The curcumin analogs were obtained from a literature search ( Pabon, 1964 ; Ohtsu et al, 2003 ; Robinson et al, 2003 , 2005 ; Nichols et al, 2006 ; Ohori et al, 2006 ; Simoni et al, 2008 ; Basile et al, 2009 ; Xiao et al, 2010 ; Kudo et al, 2011 ; Sreenivasan et al, 2013 ; Ahn et al, 2014 ; Rampogu et al, 2022 ). The chalcone analogs/derivatives were retrieved from several literature sources ( Boeck et al, 2006 ; Choudhary & Juyal, 2011 ; Gupta & Jain, 2015 ; Bui et al, 2016 ; Pesaran Seiied Bonakdar et al, 2017 ; Gomes et al, 2017 ; Teng et al, 2018 ; Zhu et al, 2019 ; Higgs et al, 2019 ; Kaur, Singh & Narasimhan, 2019 ; Aljamali, Hamzah Daylee & Jaber Kadhium, 2020 ; Rammohan et al, 2020 ; Okolo et al, 2021 ; Vadivoo et al, 2021 ; Wijayanti et al, 2021 ; Konidala et al, 2021 ; Abosalim, Nael & El-Moselhy, 2021 ; Ouyang et al, 2021 ; Rampogu et al, 2021 ; Taresh, 2022 ) to build a webserver that could help in the virtual screening process.…”

Section: Methodsmentioning

confidence: 99%

Curcumin Chalcone Derivatives Database (CCDD): a Python framework for natural compound derivatives database

Rampogu,

Balasubramaniyam,

Lee

2023

PeerJ

View full text Add to dashboard Cite

We built the Curcumin Chalcone Derivatives Database (CCDD) to enable the effective virtual screening of highly potent curcumin and its analogs. The two-dimensional (2D) structures were drawn using the ChemBioOffice package and converted to 3D structures using Discovery Studio Visualizer V 2021 (DS). The database was built using different Python modules. For the 3D structures, different Python packages were used to obtain the data frame of compounds. This framework is also used to visualize the compounds. The webserver enables the users to screen the compounds according to Lipinski’s rule of five. The structures can be downloaded in .sdf and .mol format. The data frame (df) can be downloaded in .csv format. Our webserver can help computational drug discovery researchers find new therapeutics and build new webservers. The CCDD is freely available at: https://srampogu-ccdd-ccdd-8uldk8.streamlit.app/.

show abstract

Section: Methodsmentioning

confidence: 99%

Curcumin Chalcone Derivatives Database (CCDD): a Python framework for natural compound derivatives database

Rampogu,

Balasubramaniyam,

Lee

2023

PeerJ

View full text Add to dashboard Cite

show abstract

“…The structure of chalcones is a key factor that determine their biological activity. In this regard, the number and position of various substituents, mainly hydroxyl groups and the á,â-double bond are important [13]. Moreover, chalcones can be modified by the addition of specified moieties to obtain the desired activities.…”

Section: Chalcones Biological Activities and Their Applications In Ag...mentioning

confidence: 99%

“…Derivatives containing phenoxyacetic acid, 4-(N,N-dimethylamino)phenyl, Nmethylpyrrole, or especially thiophenyl functional groups have shown promising inhibitory activity. [10,13].…”

Section: Herbicides and Plant Growth Regulatorsmentioning

confidence: 99%

“…Interestingly, a single compound may exibit several activities, for example isobavachalcone is known to have chemopreventive, anti-cancer, anti-bacterial and anti-fungal activities [11,12]. Naturally occurring chalcones have been used in traditional medicine for years, only now new applications appear [13]. Due to increased effort to reduce synthetic pesticides usage within Farm to Fork strategy from the European Union until 2030, biopesticides are gaining popularity not only because of different mode of action but also, and more importantly, they are more environmentally friendly.…”

Section: Introductionmentioning

confidence: 99%

See 1 more Smart Citation

Chalcones – Features, Identification Techniques, Attributes and Application in Agriculture

Dziągwa-Becker,

Oleszek,

Zielińska

et al. 2024

Preprint

View full text Add to dashboard Cite

This review provides a comprehensive and updated information on chalcones, presenting their sources, methods of identification and properties putting emphasis on applications in agricultural industry. Vast exploitation of synthetic pesticides led to the weed and pest resistance issue, causing economic loss but more importantly health risk due to pesticide overuse. Because one of the aim of the European Green Deal 2030 is the Farm to Fork strategy which targets on reducing by 50% the use of chemical pesticides by 2030, and push towards natural pesticides which are more environmentally friendly and restore natural resources, chalcones and their derivatives seem to fit perfectly. They have herbicidal, fungicidal, bactericidal and antiviral properties. Moreover, chalcones are naturally occurring substances, known for their favorable health effect for years, working on many areas. This review is complementary to the previous ones describing chalcones use in agriculture, updates them but additionally shows methods of detection.

show abstract

“…6 Antipyrine is a lowtoxicity drug that was first prepared by Connor in 1883 AD. 7,8 Benzothiazoles are bicyclic compounds that are heterocyclic organic compounds containing a benzene ring attached to a five-membered thiazole ring containing nitrogen and sulfur atoms. 9 It is a weak base and is a colorless and slightly viscous liquid with a melting point of (2°C), boiling point (227-228°C) and is slightly soluble in water.…”

mentioning

confidence: 99%

Synthesis, Characterization of New Ligand Derived from 4-aminoantipyrine and its Complexes with Few Metallic Ions and Evaluation of their Activity as Anticancer

Dawood¹,

Jamel²

2022

IJDDT

View full text Add to dashboard Cite

A new heterocyclic ligand (LH) derived from 4-aminoantipyrene was prepared through the reaction of 2-mercaptobenzothiazole with 4-amino-antipyrene dissolved in absolute ethanol as the first step to form compound-A, while the second step involved the reaction of O-phenylenediamine with benzil to produce compound -B, the third step involved the reaction of the products of the first and second steps to give the ligand as a final product. Five complexes, Ni (II), Cu (II), Zn(II), Cd (II) and Ag (I) were synthesized from the reaction of the ligand (LH) with its ionic salts. The ligand and its prepared complexes are characterized by proton nuclear magnetic resonance (1H-NMR), fourier-transform infrared spectroscopy (FTIR), UV-vis spectroscopy and X-rays as well as used other techniques such as quantitative analysis of the elements china health and nutrition survey (CHNS), field emission scanning electron microscope (FESEM) as well as molar conductivity and magnetism sensitivity, in addition to measuring melting points. These techniques were used to determine the structures and geometry of the prepared compounds. FTIR spectra showed that the ligand behaves as a tetra-dentate ligand and that the ratio of ligand to metal is (1:1) for all the prepared complexes according to the molar ratio calculations, which were confirmed by quantitative analysis of the elements CHNS and atomic absorption measurements. The molar conductivity results showed that all the non-electrolytic complexes except the zinc (II) and cadmium (II) complexes were ionic in a 1:1 ratio. From the foregoing, it is proved that the complexes have tetrahedral geometry, with the exception of the Ni(II) and Cu(II) complexes, which are octahedral. The anticancer activity of the ligand and its complex with silver was further evaluated using breast cancer cell lines and compared to the normal cell line. The study showed good results by treating infected cells compared to normal cells.

show abstract

A Literature Review on Antipyrinein Chemistry Fields

Cited by 6 publications

References 24 publications

Curcumin Chalcone Derivatives Database (CCDD): a Python framework for natural compound derivatives database

Curcumin Chalcone Derivatives Database (CCDD): a Python framework for natural compound derivatives database

Chalcones – Features, Identification Techniques, Attributes and Application in Agriculture

Synthesis, Characterization of New Ligand Derived from 4-aminoantipyrine and its Complexes with Few Metallic Ions and Evaluation of their Activity as Anticancer

Contact Info

Product

Resources

About