Weak-coordination-auxiliary aminocatalysis enables directed [3 + 2] cyclization for 2-acylindolizines
Kui Zeng,
Neeraj Kumar Pandit,
João C. A. Oliveira
et al.
Abstract:The synthesis of 2-acylindolizines, possessing a readily modifiable ketone group, is of significant importance as it provides versatile precursors for the preparation of various indolizines. However, due to the electronically...
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