“…- Substrates cordycepin [40], zebularine [40], tubercidin [40], cladribine [40], fludarabine [40], zalcitabine [40], didanosine [40], floxuridine [40], zidovudine [40] tetraethylammonium [194,730], MPP + [194,730], metformin [807], atenolol [486] Endogenous substrates adenosine [40], inosine [40], uridine [40], guanosine [40], thymidine [40], adenine [40] dopamine [194,730], 5-hydroxytryptamine [194,730], histamine [194,730], tyramine [194,730], adenosine [806] Stoichiometry Equilibrative Equilibrative Inhibitors -decynium 22 (pK i 7) [194,730], rhodamine123 (pK i 6) [194,730], dipyridamole (pK i 5.9) [726], verapamil (pK i 4.7) [194,730], fluoxetine (pK i 4.6) [194,730], quinidine (pK i 4.6) [194,730], quinine (pK i 4.6) [194,730], desipramine (pK i 4.5) [194,730], cimetidine (pK i <3.3) …”