Synthesis of Potential Purinoceptor Antagonists: Application of P1‐tBu Phosphazene Base for Alkylation of Adenine in Solution and on Solid Phase.

Abstract

The selective N-alkylation to the intermediates such as (V) is the key step in the synthesis of the title compounds. -(ENKVIST, E.; RAIDARU, G.; URI*, A.; PATEL, R.; REDICK, C.; BOYER, J. L.; SUBBI, J.; TAMMISTE, I.; Nucleosides, Nucleotides