Synthesis and Antiradical and Antibacterial Activity of 4-(3′,4′-Dihydroxyphenyl)Thiazole Derivatives

Odaryuk, V. V.; Burakov, N. I.; Kanibolotskaya, L. V.; Kanibolotskii, A. L.; Odaryuk, I. D.; Lebedeva, N. Yu.; Poddubnaya, E. N.; Shendrik, A. N.

doi:10.1007/s11094-015-1229-5

Cited by 3 publications

(2 citation statements)

References 5 publications

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“…Odaryuk et al designed dihydroxyphenylthiazoles series from the reaction of 4‐(chloroacetyl)catechol with thioamide derivatives. Antimicrobial activity against E. coli , Enterobacter cloacae , K. pneumoniae , P. aeruginosa , St. aureus , St. epidermidis and C. albicans was assessed for dihydroxyphenylthiazoles.…”

Section: Introductionmentioning

confidence: 99%

A retrospect on antimicrobial potential of thiazole scaffold

Mishra

Mujwar

et al. 2020

Journal of Heterocyclic Chem

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Due to its appreciable diversity in biological actions, thiazole and its substituted components, a significant class of heterocyclic compounds has developed as an influential scaffold in the field of chemical sciences. The variability of thiazole core has been expressed through the effective instigation of its anticancer (Dasatinib, Tiazofurin), antiretroviral (Ritonavir, Brecanavir), antimicrobial (Sulfathiazole, Ravuconazole) and anti-inflammatory (Fenclozic acid, Meloxicam) derivatives. This reasonable diversity in the physiological reaction pattern led many scientists to refine and develop new structural alternatives with much more efficient pharmacological action. This review is crucial for previous studies and projects to survey the antimicrobial activity of thiazole and thiazole related compounds to the mid of 2019.

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Section: Introductionmentioning

confidence: 99%

A retrospect on antimicrobial potential of thiazole scaffold

Mishra

Mujwar

et al. 2020

Journal of Heterocyclic Chem

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“…Similarly, monosubstituted thiourea 19 reacted with phenacyl chloride 18 to afford substituted 2-aminothiazole derivatives (Scheme 5). 20 showed antimicrobial activity against P. aeruginosa, S. aureus, S. epidermidis and C. albicans but it was found inactive against E. coli, E. cloacae and K. pneumoniae 23. Scheme 5.…”

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confidence: 99%

Synthetic Approaches toward Certain Structurally Related Antimicrobial Thiazole Derivatives (2010-2020)

Abuo‐Rahma¹,

Hassan²,

Hassan³

et al. 2021

HETEROCYCLES

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In the present literature review, we comprehensively discuss different methods of synthesis of published antimicrobial thiazole derivatives in the last decade mainly those which showed antibacterial, antimycobacterial and/or antifungal activity. Owing to the great diversity of thiazole-derived antimicrobial agents, we organized most of them chemically in stipulated classes. In each class, we mentioned common methods of thiazole ring closure and indicated antimicrobial activity of the most active derivatives in clear and simple way. CONTENTS1.

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