Stereochemical optimization of <i>N</i>,2-substituted cycloalkylamines as norepinephrine reuptake inhibitors

Dilweg, Majlen A.; Mocking, Tamara A. M.; Maragkoudakis, Pantelis; van Westen, Gerard J. P.; Heitman, Laura H.; IJzerman, Adriaan P.; Jespers, Willem; van der Es, Daan

doi:10.1039/d4md00521j

RSC Med. Chem.

2024

DOI: 10.1039/d4md00521j

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Stereochemical optimization of N,2-substituted cycloalkylamines as norepinephrine reuptake inhibitors

Majlen A. Dilweg,

Tamara A. M. Mocking,

Pantelis Maragkoudakis

et al.

Abstract: The norepinephrine transporter (NET), encoded by the SLC6A2 gene, is one of three key monoamine neurotransmitter transporters. Inhibition of NET-mediated reuptake of norepinephrine by monoamine reuptake inhibitors has been the...

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Stereochemical optimization of N,2-substituted cycloalkylamines as norepinephrine reuptake inhibitors

Abstract: The norepinephrine transporter (NET), encoded by the SLC6A2 gene, is one of three key monoamine neurotransmitter transporters. Inhibition of NET-mediated reuptake of norepinephrine by monoamine reuptake inhibitors has been the...

Cited by 0 publications

References 49 publications

No citations

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