N-Aryl-2-dialkylaminosuccinimides

Kolyamshin, O. A.; Danilov, V. A.

doi:10.1023/b:rujo.0000045189.81688.f3

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2024

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Cited by 6 publications

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Conjugate Additions of Amines to Maleimides via Cooperative Catalysis

et al. 2018

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A cooperative system comprising of a lithium Lewis acid and amine base significantly enhances the rate of the conjugate addition of a wide array of amines to maleimides. This operationally simple, scalable method provides mono‐addition products in high yields and purity. This conjugation was successfully applied to the kinase inhibitor crizotinib in a chemoselective ligation to create novel fluorescent probe.magnified image

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Conjugate Additions of Amines to Maleimides via Cooperative Catalysis

et al. 2018

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N‐Aryl‐2‐dialkylaminosuccinimides.

Kolyamshin

Danilov

2005

ChemInform

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Pyrrole derivatives R 0120 N-Aryl-2-dialkylaminosuccinimides. -A simple and efficient synthesis of pharmacologically interesting title compounds (III) is carried out by heating the mixture of equimolar amounts of N-arylmaleimides (I) with amines (II) in dioxane. -(KOLYAMSHIN, O. A.; DANILOV, V. A.; Russ. J. Org. Chem. 40 (2004) 7, 982-985; Chuvash Ul'yanov State Univ., Cheboksary 428015, Russia; Eng.) -R. Staver 09-099

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Microwave‐Assisted Catalyst‐Free Conjugate Addition of Amines to Maleimide

Bharodiya,

Desai,

Desai

et al. 2024

ChemistrySelect

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A catalyst‐free approach has been introduced for the conjugate addition of aromatic amine nucleophiles to α, β‐unsaturated N‐methyl maleimide under microwave irradiation by utilizing water as a promoter. Catalyst‐free, environmentally friendly, short‐reaction time, green solvent, and mild reaction conditions are the advantages of this protocol. This reaction provided good to excellent yields with aromatic anilines as nucleophiles. The benefits of this reaction align with the principles of green and sustainable synthetic chemistry, making it widely applicable in organic synthesis and pharmaceutical chemistry.

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N-Aryl-2-dialkylaminosuccinimides

Cited by 6 publications

References 1 publication

Conjugate Additions of Amines to Maleimides via Cooperative Catalysis

Conjugate Additions of Amines to Maleimides via Cooperative Catalysis

N‐Aryl‐2‐dialkylaminosuccinimides.

Microwave‐Assisted Catalyst‐Free Conjugate Addition of Amines to Maleimide

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