Isatin-3-anils as excystment and cysticidal agents againstSchizopyrenus russelli

Abstract

A series of isatin-3-anils (with or without a N-piperidino/morpholinomethyl substituent) have been screened for their cysticidal activity against Schizopyrenus russelli. Their ability to cause excystment has also been studied.

Aza‐Michael Addition of Isatin and Phthalimide to Symmetrical Fumaric Esters in Ionic Liquid Media

“…5,6 Derivatives of this compound have been also reported to possess biological activities. 7 Schiff bases and Mannich bases of isatin have antibacterial, [8][9][10] antifungal, [11][12][13] antiviral, [14][15][16] anti-HIV, [17][18][19] antiprotozoal, 20,21 and antihelminthic properties. 22,23 Isatin and its derivatives are also versatile starting materials for the synthesis of heterocyclic, non-cyclic and natural products.…”

Synthesis and antimicrobial activities of 1-(5-substituted-2-oxo indolin-3-ylidene)-4-(substituted pyridin-2-yl) thiosemicarbazide

“…1,2 Schiff bases of isatin (indolin-2,3-dione) derivatives are reported to show variety of biological activities like antibacterial, [3][4][5] antifungal, 6-8 antiviral, [9][10][11] anti HIV, [12][13][14] antiprotozoal 15,16 and antihelminthic 17,18 activities. In addition pyridines are associated with diverse biological activities.…”

One-pot rapid and efficient synthesis of new spiro derivatives of 11H-indeno[1,2-b]quinoxalin-11-one, 6H-indeno[1,2-b]pyrido[3,2-e]pyrazin-6-one and isatin-based 2-pyrazolines

“…Isatin has anxiogenic, 23 anticonvulsant 24 activity and acts as a potent antagonist on atrial natriuretic peptide receptors in vitro. 25 Isatin derivatives of Mannich bases had antibacterial, [26][27][28] antifungal, [29][30][31] antiviral, [32][33][34] anti HIV, [35][36][37] antiprotozoal, 38,39 anticancer, 40 muscle relaxant, 41 antiallergic 42 activity.…”