Influence du cytochrome P450 2D6 sur le métabolisme de la TFMPP (1-(3-trifluoro-méthylphenyl) pipérazine) : étude à l'aide de modèles in vitro et in vivo
Abstract:RÉSUMÉ
La connaissance des isoenzymes du cytochrome P450 (CYP), qui sont responsables du métabolisme des xénobiotiques, est indispensable pour prédire la toxicocinétique et Vévaluation des risques toxicologiques,
MOTS-CLÉS : l-(3-trifluoro-méthyl-phényl)pipérazine, TFMPP, métabolis-me, cytochrome P450. rats Wistar, rats Dark Agouti.
SUMMARY
Knowledge of the cytochrome P450 (CYP) isoenzymes responsible for the metabolism of xenobiotics is indispensable for prediction of toxicokinetics and for risk assessment. … Show more
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