Heteroaromatization with 4-phenyldiazenyl-1-naphthol. Part I: Synthesis of some new naphthopyrans and naphthopyranopyrimidines

Heteroaromatization of Coumarin Part I: Design, Synthesis, Re-Actions, Antitumor Activities of Novel of Chromen-3-Yl-Pyridine and Chromen-3-Yl-Naphthyridine Derivatives

“…In continuation of our research program on the synthesis of novel heterocyclic compounds exhibiting antitumor activities [15][16][17][18][19][20][21][22][23][24][25][26][27], we attempted to design pyrimidine, tetrazole and triazolopyrimidine to position 3 of coumarin as a novel 3-heteroarylcoumarins, which have not been reported hitherto, to evaluate their in vitro antitumor activity against Human breast cancer cell line (MCF-7), human cervical cancer cell line (HeLa), and human prostate cancer (PC-3).…”

New chloroamide-steroid derivative with biological activity on a casein kinase 2 (CK2)

“…Several azahexacyclo analogs have been using different methods which use some reagents such an oligoether derivative [30] [32], benzyl amine [33], thiourea/hydrochloric acid [34], α-cyanocinnamonitriles [35] and others. However, some of these reagents are expensive and require special conditions for their management.…”

Benzo[ f ]chromene Derivatives as Cytotoxic Agents: Design, Synthesis, Molecular Docking, and ADMET

“…This study builds upon our ongoing efforts to design and develop potent benzochromene-based scaffolds, specifically benzochromenes, benzochromenopyrimidines, and benzochromenotriazolopyrimidines, as potential anticancer agents. − …”