Efficient Synthesis of Chiral 1,1′‐Sulfonyl Bisaziridines

Khettache, Nawel; Bendjeddou, Amel; Berredjem, Malika; Régaı̈nia, Zine; Montero, Veronique; Menut, Chantal; Aouf, Nour‐Eddine; Winum, Jean‐Yves

doi:10.1080/00397910600639802

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Inorganic Industrial and Analytical Studies1

Alicyclic Sulfamides1

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Cited by 5 publications

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“…934 Some bisaziridine sulfamides 395 (R = Bn, iPr, and iBu) have been prepared in ∼90% yields starting from N,N′-[(NHCH 2 (R)-CO 2 Me)] 2 SO 2 . 935 Certain types of tetraarylsulfamides can be prepared generally in ≥70% yields by reaction of arylsulfamoyl imidazolium triflates such as 396, which are readily prepared from the corresponding chlorides with amines. One of the arylsulfamides made by this method is a bioisostere of the drug muraglitazar, which is in clinical development for treating type 2 diabetes and dyslipidemia.…”

Section: Inorganic Industrial and Analytical Studiesmentioning

confidence: 99%

“…Some bisaziridine sulfamides 395 (R = Bn, i Pr, and i Bu) have been prepared in ∼90% yields starting from N , N ′-[(NHCH 2 (R)CO 2 Me)] 2 SO 2 . Certain types of tetraarylsulfamides can be prepared generally in ≥70% yields by reaction of arylsulfamoyl imidazolium triflates such as 396 , which are readily prepared from the corresponding chlorides with amines.…”

Section: Alicyclic Sulfamidesmentioning

confidence: 99%

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