Eaton's reagent is an alternative of PPA: Solvent free synthesis, molecular docking and ADME studies of new angular and linear carbazole based naphtho naphthyridines

Kolandaivel, P.; Satheeshkumar, Rajendran; Aathi, Muthu Sankar; Chandrasekar, Chinnarasu; Sukantha, Tiruchengode Arumugam; Gnanamangai, Balasubramanian Mythili; Acevedo, R.; Sayın, Koray; Prasad, K. J. Rajendra

doi:10.1016/j.tet.2023.133320

Tetrahedron

2023

DOI: 10.1016/j.tet.2023.133320

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Eaton's reagent is an alternative of PPA: Solvent free synthesis, molecular docking and ADME studies of new angular and linear carbazole based naphtho naphthyridines

P. Kolandaivel¹,

Rajendran Satheeshkumar

Muthu Sankar Aathi

et al.

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2024

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Direct Synthesis of 3‐Arylphthalides Promoted by Eaton's reagent

Eddebbarh,

Moutardier,

Thibonnet

et al. 2024

Eur J Org Chem

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A rapid method has been developed for the synthesis of 3‐arylphthalides from readily available starting materials. We describe herein a direct approach based on a simple Friedel‐Crafts condensation between an aromatic ester and an aldehyde promoted by a mixture of phosphorus pentoxide and methanesulfonic acid (Eaton’s reagent) under metal and solvent‐free conditions. Due to their similarity to cytosporone E (a natural antibacterial phthalide), some of the synthesized compounds were tested as antibacterial agents against methicillin‐resistant strain of Staphylococcus aureus.

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Direct Synthesis of 3‐Arylphthalides Promoted by Eaton's reagent

Eddebbarh,

Moutardier,

Thibonnet

et al. 2024

Eur J Org Chem

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show abstract

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Eaton's reagent is an alternative of PPA: Solvent free synthesis, molecular docking and ADME studies of new angular and linear carbazole based naphtho naphthyridines

Cited by 1 publication

References 50 publications

Direct Synthesis of 3‐Arylphthalides Promoted by Eaton's reagent

Direct Synthesis of 3‐Arylphthalides Promoted by Eaton's reagent

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