ChemInform Abstract: Palladium‐Catalyzed Route to Three‐Component, One‐Pot Sequential Synthesis of Functionalized Cyclazines: 2,2a¹,4‐Triazacyclopenta[cd]indenes.

Abstract

Palladium-Catalyzed Route to Three-Component, One-Pot Sequential Synthesis of Functionalized Cyclazines: 2,2a 1 ,4-Triazacyclopenta[cd]indenes. -The synthesis of cyclazines involves initial three-component condensation and a Pd-catalyzed intramolecular α-arylation of an α-aminocarbonyl functionality. -(YANG, A.; JIANG, R.; KHOREV, O.; YU, T.; ZHANG, Y.; MA, L.; CHEN, G.; SHEN*, J.; MENG, T.; Adv. Synth. Catal. 355 (2013) 10, 1984-1988, http://dx.