Abstract:Organocatalytic Entry into 2,6-Disubstituted Aza-Achmatowicz Piperidinones: Application to (-)-Sedacryptine and Its Epimer. -(-)-Sedacryptine (XIII) and its epimer (XVI) are prepared via organocatalyzed Mannich, aza-Achmatowicz, and an N-acyliminium ion addition reaction from boc-protected furanyl amines. -(VAN DER PIJL, F.; HARMEL, R. K.; RICHELLE, G. J. J.; JANSSEN, P.; VAN DELFT, F. L.; RUTJES*, F. P. J. T.; Org. Lett. 16 (2014) 7, 2038-2041, http://dx.doi.org/10.1021/ol500633u ; Inst. Mol. Mater., Radboud … Show more
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