ChemInform Abstract: Hypervalent Iodine Mediated One‐Pot C‐H Functionalization at 2α‐ or 3α‐Position of Indole Derivatives.

Abstract

The hypervalent iodine-mediated one-pot C-H functionalization at the 2-or 3-position of indole derivatives is studied. Ph-I(N 3)2 needed for the introduction of the azido group can be prepared in situ from iodosobenzene and trimethylsilylazide. -(HIGUCHI, K.; KAWASAKI*, T.; INABA, M.; NAGANUMA, A.; ISHIZAKI, T.; TAYU, M.; Heterocycles 89 (2014) 9, 2105-2121, http://dx.doi.org/10.3987/COM-14-13065 ; Meiji Pharm. Univ., Kiyose, Tokyo 204, Japan; Eng.) -M. Bohle 09-152