Abstract:Malaria masih lagi kekal menjadi salah satu penyakit endemik yang boleh membawa maut dan rawatan yang digunakan kini untuk merawat malaria adalah terapi gabungan artemisinin. Namun begitu, akses kepada rawatan ini adalah sangat terhad dan memberi kesan besar kepada negara miskin disebabkan kos terapi yang tinggi. Penilaian aktiviti antimalaria bagi kompleks organologam berasaskan ligan makroksiklik tetraaza masih kurang meluas dijalankan. Ligan makrosiklik tetraaza 5,5,7,12,12,14- heksametil-1,4,8,11- tetraaza… Show more
“…The higher SI value (SI > 10) for a test compound theoretically indicates the effectiveness and safety of a drug. [50][51][52][53] Molecular docking…”
Research on the antimalarial effect of aminoalkyl chalcone derivatives against Plasmodium falciparum and Plasmodium knowlesi has bolstered efforts in drug discovery to combat cases of drug resistance.
“…The higher SI value (SI > 10) for a test compound theoretically indicates the effectiveness and safety of a drug. [50][51][52][53] Molecular docking…”
Research on the antimalarial effect of aminoalkyl chalcone derivatives against Plasmodium falciparum and Plasmodium knowlesi has bolstered efforts in drug discovery to combat cases of drug resistance.
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