acetamido]thio-4H-1,2,4-triazole Derivatives. -Triazoles incorporating a thiazole ring system, and additionally in some cases an ester residue, are synthesized and evaluated for antifungal and antibactrial activity. Five triazolinethiones (V) and fifteen new thioether derivatives of (V) are prepared. Thiotriazoles are more active than their thioether derivatives, especially the tolyloxy derivatives (Vb) and (Ve), the triazoles are more active towards fungi than bacteria. The antibacterial assessment reveals only a slight or moderate activity. -(TURAN-ZITOUNI*, G.; KAPLANCIKLI, Z. A.; YILDIZ, M. T.; CHEVALLET, P.; KAYA, D.; Eur. J. Med. Chem. 40 (2005) 6, 607-613; Dep. Pharm. Chem., Fac. Pharm., Anadolu Univ., TR-26470 Eskisehir, Turk.; Eng.) -H. Hoennerscheid 42-147
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