Design and Synthesis of Polycyclic Acridin-(9-yl-Amino)Thiazol-5-yl)-2H-Chromen-2-One Derivatives: As Antiproliferative and Anti-TB Pharmacophores

Mane, Smita; Katagi, Kariyappa S.; Kadam, Nikhil S.; Akki, Mahesh; Joshi, Shrinivas D.

doi:10.1080/10406638.2020.1734636

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Coumarin Hybrids1

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2024

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Cited by 2 publications

(1 citation statement)

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“…A series of nine novel acridine–thiazole bridged coumarin derivatives was prepared and evaluated for their in vitro antiproliferative activity on MDA-MB-231, A-549, and HT29 cell lines. 99 All the compounds showed a significant cytotoxicity effect but none of them were more potent than the reference cisplatin. Compound 53a ( Fig.…”

Section: Coumarin Hybridsmentioning

confidence: 95%

Latest developments in coumarin-based anticancer agents: mechanism of action and structure–activity relationship studies

Koley,

Han,

Soloshonok

et al. 2024

RSC Med. Chem.

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Section: Coumarin Hybridsmentioning

confidence: 95%

Latest developments in coumarin-based anticancer agents: mechanism of action and structure–activity relationship studies

Koley,

Han,

Soloshonok

et al. 2024

RSC Med. Chem.

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Recent Literature on the Synthesis of Thiazole Derivatives and their Biological Activities

Farghaly

Alfaifi

Gomha

2024

MRMC

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The thiazole ring is naturally occurring and is primarily found in marine and microbial sources. It has been identified in various compounds such as peptides, vitamins (thiamine), alkaloids, epothilone, and chlorophyll. Thiazole-containing compounds are widely recognized for their antibacterial, antifungal, anti-inflammatory, antimalarial, antitubercular, antidiabetic, antioxidant, anticonvulsant, anticancer, and cardiovascular activities. The objective of this review is to present recent advancements in the discovery of biologically active thiazole derivatives, including their synthetic methods and biological effects. This review comprehensively discusses the synthesis methods of thiazole and its corresponding biological activities within a specific timeframe, from 2017 until the conclusion of 2022.

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Design and Synthesis of Polycyclic Acridin-(9-yl-Amino)Thiazol-5-yl)-2H-Chromen-2-One Derivatives: As Antiproliferative and Anti-TB Pharmacophores

Cited by 2 publications

References 26 publications

Latest developments in coumarin-based anticancer agents: mechanism of action and structure–activity relationship studies

Latest developments in coumarin-based anticancer agents: mechanism of action and structure–activity relationship studies

Recent Literature on the Synthesis of Thiazole Derivatives and their Biological Activities

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